SCHEMBL8883103

SCHEMBL8883103

O=C(O)c1ncccc1OCCCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASPH Q12797 3/20 0.49
KDM8 Q8N371 3/20 0.49
LMNA P02545 1/20 0.47
IDO1 P14902 1/20 0.47
CYP11B1 P15538 3/20 0.47
CYP11B2 P19099 3/20 0.47
FFAR1 O14842 1/20 0.47
KDM4E B2RXH2 3/20 0.45
MAPT P10636 2/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
BLM P54132 1/20 0.45
AGER Q15109 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8882396 0.95 ASPH (0.50) ASPHKDM8CYP11B1CYP11B2FFAR1
SCHEMBL8883428 0.92 CYP11B1 (0.55) ASPHKDM8IDO1CYP11B1CYP11B2
SCHEMBL2426791 0.83 LTA4H (0.58) KDM4EALDH1A1
SCHEMBL30848623 0.83 LTA4H (0.58) KDM4EALDH1A1
SCHEMBL21248064 0.82 ALDH1A1 (0.49) LMNAKDM4EMAPTALDH1A1CYP3A4
SCHEMBL12697756 0.81 KDM4E (0.50) LMNAKDM4EMAPTALDH1A1CYP3A4
SCHEMBL8881039 0.81 PTPN1 (0.55) LMNAKDM4EMAPTALDH1A1CYP3A4
Hydrochloric Acid SCHEMBL10705444 0.81 LTA4H (0.57) KDM4EALDH1A1
SCHEMBL1138239 0.81 KDM4E (0.50) KDM4EMAPTALDH1A1CYP3A4ALOX15
SCHEMBL6042801 0.80 PTPN1 (0.51) LMNAKDM4EMAPTALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658933-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AKTIENGESELLSCHAFT (DE) 1997-08-19 US disclosed
CN-1107144-A Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1995-08-23 CN disclosed
CN-1107145-A Substituted heterocyclic carboxamides, their preparation and their use as pharmaceuticals HOECHST AG (DE) 1995-08-23 CN disclosed