SCHEMBL8889786

SCHEMBL8889786

O=c1ccc(-c2c(-c3cccc(Cl)c3)n[nH]c2-c2cccc(Cl)c2)n[nH]1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
AKR1B1 P15121 1/20 0.42
NOTUM Q6P988 1/20 0.42
HPGD P15428 1/20 0.41
HTR7 P34969 1/20 0.40
AHR P35869 1/20 0.40
ATM Q13315 1/20 0.40
GRM5 P41594 2/20 0.39
MET P08581 1/20 0.39
PDGFRB P09619 1/20 0.39
CDK8 P49336 1/20 0.39
ROCK1 Q13464 1/20 0.39
NTRK3 Q16288 1/20 0.39
NTRK2 Q16620 1/20 0.39
AURKB Q96GD4 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
IDO1 P14902 3/20 0.39
IKBKE Q14164 1/20 0.38
TGFBR1 P36897 1/20 0.38
TGFBR2 P37173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888361 0.95 CYP1A2 (0.50) CYP1A2AKR1B1NOTUMHPGDHTR7
SCHEMBL8889484 0.87 CYP1A2 (0.53) CYP1A2AKR1B1HPGDGRM5IDO1
SCHEMBL8888295 0.82 CYP1A2 (0.53) CYP1A2HPGDATMGRM5MAPK11
SCHEMBL4048920 0.81 CYP1A2 (0.62) CYP1A2AKR1B1NOTUMAHRIDO1
Bromide SCHEMBL11739258 0.80 CYP1A2 (0.61) CYP1A2AKR1B1NOTUMAHRIDO1
SCHEMBL8887885 0.80 CYP1A2 (0.50) CYP1A2NOTUMHPGDHTR7IDO1
SCHEMBL8890194 0.80 CYP1A2 (0.50) CYP1A2HPGDMAPK11MAPK14GPR119
SCHEMBL8887621 0.80 CYP1A2 (0.50) CYP1A2NOTUMHPGDHTR7MAPK14
SCHEMBL8889663 0.77 CYP1A2 (0.47) CYP1A2AKR1B1NOTUMHPGDIDO1
SCHEMBL8886941 0.77 NR1H2 (0.49) CYP1A2NOTUMHPGDMAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed