SCHEMBL8887885

SCHEMBL8887885

O=c1ccc(-c2c(-c3cccc(F)c3)n[nH]c2-c2ccccc2)n[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
MAPK13 O15264 1/20 0.43
RAF1 P04049 1/20 0.43
MAPK12 P53778 1/20 0.43
MAPK11 Q15759 1/20 0.43
MAPK14 Q16539 1/20 0.43
GPR119 Q8TDV5 1/20 0.41
NOTUM Q6P988 1/20 0.40
HPGD P15428 2/20 0.40
MAPK1 P28482 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888361 0.85 CYP1A2 (0.50) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8890194 0.85 CYP1A2 (0.50) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8887621 0.85 CYP1A2 (0.50) CYP1A2MAPK14GPR119NOTUMHPGD
SCHEMBL8897726 0.82 JAK2 (0.46) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8889484 0.82 CYP1A2 (0.53) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8889663 0.82 CYP1A2 (0.47) CYP1A2GPR119NOTUMHPGDSMN1; SMN2
SCHEMBL8886941 0.82 NR1H2 (0.49) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8888926 0.80 KMT2A (0.57) CYP1A2GPR119HPGDMAPK1SMN1; SMN2
SCHEMBL8888295 0.80 CYP1A2 (0.53) CYP1A2MAPK13RAF1MAPK12MAPK11
SCHEMBL8889786 0.80 CYP1A2 (0.45) CYP1A2MAPK11MAPK14GPR119NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997001551-A1 PYRAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-01-16 WO disclosed