SCHEMBL8891765

SCHEMBL8891765

Cc1cc2c(cc1C#Cc1ccc(C(=O)O)cn1)C(C)(C)CC(C)(C)O2

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
CYP26A1 O43174 1/20 0.46
RXRA P19793 7/20 0.39
RARB P10826 5/20 0.39
RARG P13631 5/20 0.39
RXRB P28702 5/20 0.39
RXRG P48443 5/20 0.39
RARA P10276 4/20 0.39
PPARG P37231 1/20 0.39
KMT2A Q03164 1/20 0.38
SLC16A3 O15427 1/20 0.36
SSTR5 P35346 1/20 0.35
GRM5 P41594 5/20 0.34
AKR1B1 P15121 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8560124 0.88 RARA (0.52) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8874667 0.85 CYP26A1 (0.40) CYP3A4CYP26A1RXRARARBRARG
SCHEMBL9180450 0.84 RARB (0.48) CYP3A4CYP26A1RXRARARBRARG
SCHEMBL8890751 0.83 CYP3A4 (0.59) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL9318320 0.82 RXRA (0.58) CYP3A4CYP26A1RXRARARBRARG
SCHEMBL8890799 0.81 GABRP (0.36) SSTR5AKR1B1
SCHEMBL8865618 0.80 CYP3A4 (0.39) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8875462 0.80 AKR1B1 (0.36) CYP26A1AKR1B1
SCHEMBL8865958 0.80 RARA (0.51) CYP3A4CYP26A1RARBRARGRARA
SCHEMBL8890100 0.80 CYP3A4 (0.52) CYP3A4CYP26A1RXRARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616597-A ANTIACNE, ANTIPSORIASIS COMPOUNDS ALLERGAN (US) 1997-04-01 US disclosed
US-5272156-A Acetylenes disubstituted with a heteroaromatic group and a 2-substituted 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1993-12-21 US disclosed
US-5045551-A Acetylenes disubstituted with a heteroaromatic group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1991-09-03 US disclosed