SCHEMBL8890954

SCHEMBL8890954

O=C1c2cc(O)ccc2CCC1Cc1cccc(NS(=O)(=O)C(F)(F)F)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.53
CYP26A1 O43174 7/20 0.47
ESR1 P03372 5/20 0.43
ESR2 Q92731 5/20 0.43
CYP24A1 Q07973 1/20 0.41
MAPK14 Q16539 1/20 0.38
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TP53 P04637 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8888125 0.86 CYP19A1 (0.56) CYP19A1CYP26A1CYP24A1
SCHEMBL8900137 0.82 MAOB (0.43) ALDH1A1SMN1; SMN2TP53CYP3A4MAPT
SCHEMBL8890267 0.80 CYP19A1 (0.50) CYP19A1CYP26A1ESR1ESR2CA2
SCHEMBL8890711 0.78 LTB4R (0.40) ESR1ESR2CYP3A4CA2
SCHEMBL8890710 0.78 LTB4R (0.40) ESR1ESR2CYP3A4CA2
SCHEMBL8465475 0.78 CYP19A1 (0.78) CYP19A1CYP26A1ESR1ESR2CYP24A1
SCHEMBL8890679 0.72 CYSLTR1 (0.38) ESR1CYP3A4CYP2D6MAPTCA2
SCHEMBL7745124 0.72 CYP26A1 (0.66) CYP19A1CYP26A1ESR1ESR2CYP24A1
SCHEMBL8892969 0.70 CYSLTR2 (0.45) MAPTCA2
SCHEMBL8892971 0.70 CYSLTR2 (0.45) MAPTCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5641789-A INHIBITORS OF LEUKOTRIENES AND/OR BLOCKERS OF LEUKOTRIENE RECEPTORS; USEFUL IN PREVENTION OR TREATMENT OF ASTHMA, ARTHRITIS, PSORIASIS, ULCERS, MYOCARDIAL INFARCTION PFIZER INC. (US) 1997-06-24 US disclosed