SCHEMBL8891085

SCHEMBL8891085

CC(=O)Nc1ccc(C(=O)O)cc1-n1cc(-c2cccc(F)c2)nc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.41
TOP2A P11388 1/20 0.41
PTGFR P43088 2/20 0.40
ATR Q13535 1/20 0.39
HPGDS O60760 2/20 0.38
KMO O15229 2/20 0.38
NEU3 Q9UQ49 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
CREBBP Q92793 1/20 0.38
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
TP53 P04637 1/20 0.37
MAPT P10636 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CG P48736 1/20 0.37
HDAC1 Q13547 2/20 0.37
KDR P35968 1/20 0.37
HDAC3 O15379 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8901022 0.90 ADORA3 (0.44) PTGFRNEU3ADORA2AADORA1ADORA3
Trifluoroacetic Acid SCHEMBL8901207 0.86 ALDH1A1 (0.40) PTGFRATRNEU3ADORA2AADORA1
SCHEMBL8892711 0.85 KEAP1 (0.46) TP53MAPTHDAC2
SCHEMBL8891817 0.83 ADORA3 (0.44) NEU3ADORA3MAPT
SCHEMBL8891736 0.82 ADORA3 (0.46) NEU3ADORA3MAPTHDAC1
SCHEMBL8891755 0.82 PTGFR (0.41) PTGFRNEU3ADORA3MAPTHDAC1
Trifluoroacetic Acid SCHEMBL8902577 0.82 KEAP1 (0.42) TP53MAPTHDAC2
Trifluoroacetic Acid SCHEMBL8894608 0.80 ADORA3 (0.40) NEU3ADORA3TP53MAPTPIK3CA
Trifluoroacetic Acid SCHEMBL8891099 0.80 ADORA3 (0.41) NEU3ADORA3MAPT
SCHEMBL8892526 0.79 ADORA3 (0.47) NEU3ADORA2AADORA1ADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997033872-A1 ANTI-VIRAL 4-ACYLAMINO-3-[IMIDAZOL-I-YL]-BENZOIC ACID DERIVATIVES BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 1997-09-18 WO claimed
WO-1997033872-A1 ANTI-VIRAL 4-ACYLAMINO-3-[IMIDAZOL-I-YL]-BENZOIC ACID DERIVATIVES BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 1997-09-18 WO disclosed