SCHEMBL8891817

SCHEMBL8891817

CC(=O)Nc1ccc(C(=O)O)cc1-n1cc(-c2ccc(C)cc2)nc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.44
KDM4E B2RXH2 8/20 0.42
MAPT P10636 6/20 0.42
NPC1 O15118 5/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
GAA P10253 2/20 0.42
GFER P55789 1/20 0.42
HPGD P15428 7/20 0.41
ALDH1A1 P00352 7/20 0.41
RAB9A P51151 3/20 0.41
NEU3 Q9UQ49 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TMIGD3 P0DMS9 1/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
LMNA P02545 1/20 0.39
PDE10A Q9Y233 1/20 0.38
CTRC Q99895 1/20 0.38
POLB P06746 2/20 0.37
MAP4K4 O95819 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8894608 0.94 ADORA3 (0.40) ADORA3KDM4EMAPTNPC1SMN1; SMN2
SCHEMBL8901022 0.91 ADORA3 (0.44) ADORA3KDM4EMAPTNPC1SMN1; SMN2
SCHEMBL8891736 0.90 ADORA3 (0.46) ADORA3KDM4EMAPTNPC1SMN1; SMN2
SCHEMBL8891755 0.90 PTGFR (0.41) ADORA3KDM4EMAPTNPC1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL8901207 0.85 ALDH1A1 (0.40) ADORA3KDM4EMAPTNPC1SMN1; SMN2
SCHEMBL8892669 0.85 SCN2A (0.45) KDM4EMAPTNPC1SMN1; SMN2GAA
Trifluoroacetic Acid SCHEMBL8891099 0.85 ADORA3 (0.41) ADORA3KDM4EMAPTSMN1; SMN2HPGD
SCHEMBL8894617 0.83 ADORA3 (0.38) ADORA3KDM4EMAPTNPC1SMN1; SMN2
SCHEMBL8891085 0.83 TLR8 (0.41) ADORA3MAPTNEU3
SCHEMBL8892711 0.80 KEAP1 (0.46) KDM4EMAPTNPC1SMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997033872-A1 ANTI-VIRAL 4-ACYLAMINO-3-[IMIDAZOL-I-YL]-BENZOIC ACID DERIVATIVES BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 1997-09-18 WO claimed
WO-1997033872-A1 ANTI-VIRAL 4-ACYLAMINO-3-[IMIDAZOL-I-YL]-BENZOIC ACID DERIVATIVES BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 1997-09-18 WO disclosed