SCHEMBL8891201

SCHEMBL8891201

COc1cnc(C(=O)O)cc1OCCc1cccnc1.[N-]=[N+]=N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.45
CYP11B2 P19099 6/20 0.45
CHEK1 O14757 1/20 0.42
RECQL P46063 1/20 0.40
TRPC6 Q9Y210 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
PTAFR P25105 2/20 0.39
CYP19A1 P11511 2/20 0.39
SIGMAR1 Q99720 1/20 0.39
GCK P35557 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8890675 0.94 CYP11B1 (0.50) CYP11B1CYP11B2CHEK1RECQLTRPC6
SCHEMBL8888044 0.84 KDM4E (0.47) CYP11B1CYP11B2TRPC6L3MBTL1ALDH1A1
SCHEMBL8891050 0.84 CYP11B1 (0.47) CYP11B1CYP11B2CHEK1RECQLL3MBTL1
SCHEMBL8889269 0.82 KDM4E (0.42) CHEK1ALDH1A1NPSR1CYP1A2
SCHEMBL21045912 0.78 TRPC6 (0.57) CYP11B1CYP11B2TRPC6PDE4APDE4B
SCHEMBL8889603 0.78 ALDH1A1 (0.58) CYP11B1CYP11B2L3MBTL1PDE4APDE4B
SCHEMBL8891482 0.77 PDE4D (0.52) CYP11B1CYP11B2RECQLL3MBTL1PDE4A
SCHEMBL8891569 0.76 KDM4E (0.52) CYP11B1CYP11B2TRPC6L3MBTL1ALDH1A1
SCHEMBL8892821 0.74 KDM4E (0.47) CHEK1ALDH1A1NPSR1CYP1A2
SCHEMBL8890700 0.73 ALDH1A1 (0.57) CYP11B1CYP11B2L3MBTL1USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997003967-A1 SUBSTITUTED AROMATIC COMPOUNDS AND THEIR PHARMACEUTICAL USE RHONE-POULENC RORER LIMITED (GB) 1997-02-06 WO disclosed