SCHEMBL8892913

SCHEMBL8892913

CC(=O)Nc1ccc(C(=O)OC(=O)C(F)(F)F)cc1-n1cc(-c2ccco2)nc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.41
ADORA1 P30542 3/20 0.41
ADORA3 P0DMS8 3/20 0.41
ADORA2B P29275 2/20 0.41
CFTR P13569 2/20 0.38
PTGS1 P23219 1/20 0.38
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
HPGD P15428 3/20 0.37
HSD17B10 Q99714 4/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
ESR1 P03372 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ESR2 Q92731 1/20 0.36
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8892900 0.87 ADORA2A (0.43) ADORA2AADORA1ADORA3ADORA2BCFTR
SCHEMBL8901213 0.86 ALDH1A1 (0.38) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL8892526 0.84 ADORA3 (0.47) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL8894617 0.83 ADORA3 (0.38) ADORA3KDM4EALDH1A1HPGDKMT2A
SCHEMBL8891105 0.82 ADORA3 (0.39) ADORA3ALDH1A1KMT2AMEN1MAPT
SCHEMBL8902589 0.79 KMT2A (0.39) KDM4EALDH1A1KMT2AMEN1MAPT
SCHEMBL8901564 0.76 ALDH1A1 (0.34) ALDH1A1HPGDKMT2ALMNACYP1A2
Trifluoroacetic Acid SCHEMBL8894379 0.73 NEU3 (0.33) CFTRKDM4EALDH1A1HPGDHSD17B10
Trifluoroacetic Acid SCHEMBL8901207 0.72 ALDH1A1 (0.40) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL8900955 0.72 SCN3A (0.41) ADORA2AADORA1ADORA3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997033872-A1 ANTI-VIRAL 4-ACYLAMINO-3-[IMIDAZOL-I-YL]-BENZOIC ACID DERIVATIVES BIOTA SCIENTIFIC MANAGEMENT PTY. LTD. (AU) 1997-09-18 WO disclosed