SCHEMBL8894848

SCHEMBL8894848

COC(=O)c1ccc(CCc2ccccc2)c(S(C)(=O)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
HPGD P15428 4/20 0.47
PTGS2 P35354 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALOX15 P16050 1/20 0.47
ALOX12 P18054 1/20 0.47
CYP2C19 P33261 1/20 0.47
CKS1B P61024 1/20 0.47
SKP2 Q13309 1/20 0.47
HIF1A Q16665 1/20 0.47
HSD17B10 Q99714 1/20 0.47
VCAM1 P19320 1/20 0.47
MGLL Q99685 1/20 0.47
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
CYP4F2 P78329 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895743 0.88 PTGS2 (0.48) ALDH1A1HPGDPTGS2CYP1A2CYP3A4
SCHEMBL8917863 0.82 VCAM1 (0.55) ALDH1A1HPGDPTGS2TP53CYP1A2
SCHEMBL27652105 0.79 VCAM1 (0.52) ALDH1A1HPGDPTGS2TP53CYP1A2
SCHEMBL8334682 0.79 VCAM1 (0.47) ALDH1A1HPGDPTGS2CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL8896876 0.78 SCN2A (0.40) ALDH1A1TP53HSD17B10GAAMAPT
SCHEMBL8408482 0.78 HPGD (0.70) ALDH1A1HPGDTP53CYP1A2CYP3A4
SCHEMBL8162236 0.77 ALDH1A1 (0.60) ALDH1A1HPGDTP53CYP1A2CYP3A4
SCHEMBL20092523 0.77 NR3C1 (0.57) ALDH1A1HPGDPTGS2CYP1A2CYP2C19
SCHEMBL8816182 0.77 VCAM1 (0.50) ALDH1A1HPGDPTGS2CYP1A2CYP2C19
SCHEMBL8409498 0.77 LMNA (0.50) ALDH1A1HPGDTP53CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693672-A 3,4,5-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1997-12-02 US disclosed