SCHEMBL8894874

SCHEMBL8894874

CC(C)(C)OC(=O)N1CCC2(CC1)C(=O)N(CC(=O)O)CN2C1CCCCC1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 2/20 0.57
NPC1L1 Q9UHC9 12/20 0.50
EPHX1 P07099 1/20 0.40
HPGD P15428 1/20 0.39
DDR1 Q08345 2/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
ENPP2 Q13822 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8894056 0.84 BDKRB2 (0.59) BDKRB2NPC1L1EPHX1
SCHEMBL8892471 0.78 BDKRB2 (0.55) BDKRB2NPC1L1DDR1
SCHEMBL1855447 0.76 NPC1L1 (0.70) BDKRB2NPC1L1DDR1
SCHEMBL8897218 0.74 NPC1L1 (0.60) BDKRB2NPC1L1DDR1
SCHEMBL8894157 0.73 NPC1L1 (0.59) BDKRB2NPC1L1DDR1
SCHEMBL17149529 0.73 EPHX1 (0.43) NPC1L1EPHX1HPGDDDB1CRBN
SCHEMBL23288815 0.71 KCNH2 (0.44) NPC1L1EPHX1HPGDDDB1CRBN
SCHEMBL5134060 0.71 GRIN2B (0.49) BDKRB2NPC1L1DDR1
SCHEMBL14282652 0.69 GRIN2B (0.50) NPC1L1DDB1CRBN
SCHEMBL31537333 0.69 CTSD (0.44) EPHX1HPGDDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5610142-A Bradykinin antagonist pseudopeptide derivatives of substituted 4-keto-1,3,8-triazaspiro[4.5]decan-3-alkanoic acids SCIOS INC. (US) 1997-03-11 US disclosed