Racephenicol

Racephenicol

SCHEMBL8895477

CS(=O)(=O)c1ccc(C(O)C(CO)NC(=O)C(Cl)Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 1.00
TSHR P16473 2/20 1.00
CYP3A4 P08684 3/20 0.78
MEN1 O00255 1/20 0.78
KMT2A Q03164 1/20 0.78
RPLP1 P05386 1/20 0.65
RPLP0 P05388 1/20 0.65
RPS17 P08708 1/20 0.65
RPSA P08865 1/20 0.65
RPS2 P15880 1/20 0.65
RPL35A P18077 1/20 0.65
RPL7 P18124 1/20 0.65
RPL17 P18621 1/20 0.65
RPS4Y1 P22090 1/20 0.65
RPS3 P23396 1/20 0.65
RPS12 P25398 1/20 0.65
RPL13 P26373 1/20 0.65
RPL10 P27635 1/20 0.65
RPL12 P30050 1/20 0.65
RPL9; RPL9P7; RPL9P8; RPL9P9 P32969 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Thiamphenicol SCHEMBL34635 1.00 LMNA (1.00) LMNATSHRCYP3A4MEN1KMT2A
Racephenicol SCHEMBL30277834 1.00 LMNA (1.00) LMNATSHRCYP3A4MEN1KMT2A
Thiamphenicol SCHEMBL6245287 0.99 LMNA (0.97) LMNATSHRCYP3A4MEN1KMT2A
Florfenicol SCHEMBL3834996 0.94 LMNA (0.90) LMNATSHRCYP3A4MEN1KMT2A
Thiamphenicol SCHEMBL10380783 0.94 LMNA (0.88) LMNATSHRCYP3A4MEN1KMT2A
Thiamphenicol SCHEMBL401137 0.93 LMNA (0.86) LMNATSHRCYP3A4MEN1KMT2A
Racephenicol SCHEMBL30388685 0.92 LMNA (0.84) LMNATSHRCYP3A4MEN1KMT2A
Thiamphenicol SCHEMBL365612 0.92 LMNA (0.84) LMNATSHRCYP3A4MEN1KMT2A
Thiamphenicol SCHEMBL9295760 0.91 RPLP1 (0.83) LMNATSHRCYP3A4MEN1KMT2A
Florfenicol SCHEMBL3637832 0.88 LMNA (1.00) LMNATSHRCYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507153-B1 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORP (US) 1997-07-09 EP claimed
US-5346828-A Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase CELGENE CORPORATION (US) 1994-09-13 US claimed
EP-0507153-A2 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORPORATION (US) 1992-10-07 EP claimed
CN-119738497-A Method for detecting thiamphenicol or related substances of thiamphenicol preparation 北京四环科宝制药股份有限公司 2025-04-01 CN disclosed
EP-3607084-B1 A METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY UNIV WESTERN AUSTRALIA (AU) 2024-05-01 EP disclosed
CN-117686628-A Method for detecting thiamphenicol genotoxic impurities 江苏恒盛药业有限公司 2024-03-12 CN disclosed
US-20210292807-A1 METHOD FOR TESTING ANTIMICROBIAL SUSCEPTIBILITY THE UNIVERSITY OF WESTERN AUSTRALIA (AU) 2021-09-23 US disclosed
CN-109928901-B Synthetic method of florfenicol intermediate 上海医药工业研究院 2020-12-11 CN disclosed
EP-3718534-A1 PHARMACEUTICAL COMPOSITION CONTAINING ETHANOL AND AN ANTIBIOTIC, AND SUITABLE FOR FORMING A SOLID MASS IN CONTACT WITH A SALINE SOLUTION - ASSOCIATED PRODUCT AND DEVICE FOR CONCENTRATION AND LOCAL DELIVERY Gelnesis (FR) 2020-10-07 EP disclosed
WO-2017133517-A1 PHOSPHAMIDE DERIVATIVE, METHOD FOR MANUFACTURING THE SAME, AND USES THEREOF 四川海思科制药有限公司 2017-08-10 WO disclosed
EP-0507153-B1 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORP (US) 1997-07-09 EP disclosed
US-5346828-A Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenylpropionic acids using d-threonine aldolase CELGENE CORPORATION (US) 1994-09-13 US disclosed
EP-0507153-A2 Stereoisomeric enrichment of 2-amino-3-hydroxy-3-phenyl-propionic acids CELGENE CORPORATION (US) 1992-10-07 EP disclosed
US-4945181-A Method for resolution of racemic thiamphenicol precursors and intermediates therefor BOEHRINGER MANNHEIM GMBH (DE) 1990-07-31 US disclosed