SCHEMBL8900948

SCHEMBL8900948

O=C1C2=C(CC(C(=O)CBr)OC2)C(=O)c2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.42
SLC25A5 P05141 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
GSK3B P49841 1/20 0.33
AKR1B1 P15121 1/20 0.31
APAF1 O14727 1/20 0.31
TDP2 O95551 1/20 0.31
PRKACA P17612 1/20 0.31
CDC25B P30305 2/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
EDNRB P24530 1/20 0.30
EDNRA P25101 1/20 0.30
S100A4 P26447 1/20 0.30
GAA P10253 1/20 0.30
LMNA P02545 1/20 0.30
RAB9A P51151 1/20 0.30
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900155 0.83 AKT1 (0.47) AKT1SLC25A5SMN1; SMN2AKR1B1APAF1
SCHEMBL8902037 0.81 AKT1 (0.44) AKT1SLC25A5SMN1; SMN2APAF1TDP2
SCHEMBL8528779 0.77 AKT1 (0.42) AKT1SLC25A5SMN1; SMN2APAF1KMT2A
SCHEMBL8907639 0.74 CTH (0.38) AKT1SLC25A5SMN1; SMN2CDC25BLMNA
SCHEMBL31237790 0.73 AKT1 (0.49) AKT1SMN1; SMN2APAF1TDP2PRKACA
SCHEMBL9755756 0.71 SMN1; SMN2 (0.40) AKT1SMN1; SMN2AKR1B1KMT2AMEN1
SCHEMBL8531983 0.70 AKT1 (0.46) AKT1SMN1; SMN2APAF1TDP2CDC25B
SCHEMBL8900149 0.68 AKT1 (0.34) AKT1PRKACA
SCHEMBL8901501 0.68 HSP90AA1 (0.46) AKT1SMN1; SMN2TDP2CDC25BKMT2A
SCHEMBL8900997 0.68 HSP90AA1 (0.46) AKT1SMN1; SMN2TDP2CDC25BKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US claimed
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US disclosed