SCHEMBL8901651

SCHEMBL8901651

CCCCCCOc1nc(-c2cc(C(C)(C)C)c(O)c(C(C)(C)C)c2)nc2[nH]cnc12

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 6/20 0.38
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
PTGS2 P35354 5/20 0.36
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8902908 1.00 PTGS1 (0.38) PTGS1CDK1CCNB1PTGS2CCNA2
SCHEMBL8903449 0.88 VCAM1 (0.39) PTGS1PTGS2
SCHEMBL8903180 0.88 VCAM1 (0.39) PTGS1PTGS2
SCHEMBL8901819 0.83 PTGS2 (0.46) PTGS1PTGS2CA1CA2
SCHEMBL8901655 0.83 CDK1 (0.55) PTGS1CDK1CCNB1PTGS2CCNA2
SCHEMBL8902911 0.83 CDK1 (0.55) PTGS1CDK1CCNB1PTGS2CCNA2
SCHEMBL8902498 0.82 CDK1 (0.38) PTGS1CDK1CCNB1PTGS2CCNA2
SCHEMBL8903318 0.78 CDK1 (0.53) PTGS1CDK1CCNB1PTGS2CCNA2
SCHEMBL8902845 0.78 CA1 (0.43) PTGS1PTGS2CA1CA2
SCHEMBL8903375 0.77 RXRA (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602140-A CAUSED BY LEUKOCYTES JAPAN ENERGY CORPORATION (JP) 1997-02-11 US disclosed
EP-0675124-A2 Purine derivatives and suppressants for inflammatory diseases JAPAN ENERGY CORPORATION (JP) 1995-10-04 EP disclosed