SCHEMBL8908340

SCHEMBL8908340

NNc1ncnc(Nc2ccccc2)n1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.71
MAPT P10636 4/20 0.71
KMT2A Q03164 4/20 0.71
MEN1 O00255 3/20 0.71
KDM4E B2RXH2 1/20 0.71
BCL6 P41182 1/20 0.68
MAPK1 P28482 3/20 0.50
CDK2 P24941 3/20 0.50
IGF1R P08069 2/20 0.50
AURKA O14965 2/20 0.50
PDPK1 O15530 2/20 0.50
CDK1 P06493 2/20 0.50
LYN P07948 2/20 0.50
FGFR1 P11362 2/20 0.50
FGFR3 P22607 2/20 0.50
RPS6KB1 P23443 2/20 0.50
MARK3 P27448 2/20 0.50
RAB9A P51151 2/20 0.50
BLK P51451 2/20 0.50
RPS6KA3 P51812 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL824411 0.90 BCL6 (0.74) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL11735758 0.84 GAA (1.00) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL11797295 0.84 GAA (1.00) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL14972606 0.83 BCL6 (0.71) GAAMAPTKMT2AMEN1KDM4E
Amanozine SCHEMBL689928 0.81 BCL6 (1.00) GAAMAPTKMT2AMEN1KDM4E
Amanozine SCHEMBL30264199 0.81 BCL6 (1.00) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL11736310 0.80 GAA (0.47) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL8908228 0.79 GAA (0.81) GAAMAPTKMT2AMEN1KDM4E
Amanozine SCHEMBL2490900 0.79 BCL6 (0.96) GAAMAPTKMT2AMEN1KDM4E
SCHEMBL27617358 0.79 ADORA3 (0.67) GAAMAPTKMT2AMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188273-B2 Insecticidal (1,3,5)-triazinyl phenyl hydrazones DOW AGROSCIENCES, LLC. (US) 2012-05-29 US disclosed
US-20120040837-A1 INSECTICIDAL (1,3,5)-TRIAZINYL PHENYL HYDRAZONES DOW AGROSCIENCES LLC (US) 2012-02-16 US disclosed
US-8067588-B2 Insecticidal (1,3,5)-triazinyl phenyl hydrazones DOW AGROSCIENCES LLC (US) 2011-11-29 US disclosed
US-20090093481-A1 INSECTICIDAL (1,3,5)-TRIAZINYL PHENYL HYDRAZONES DOW AGROSCIENCES LLC (US) 2009-04-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093481-A1 INSECTICIDAL (1,3,5)-TRIAZINYL PHENYL HYDRAZONES HELZ, API5, CRYZ GAA 3359/4885MAPT 2948/4885KMT2A 1091/4885
US-20120040837-A1 INSECTICIDAL (1,3,5)-TRIAZINYL PHENYL HYDRAZONES HELZ, API5, CRYZ GAA 3359/4885MAPT 2948/4885KMT2A 1091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.