SCHEMBL8908675

SCHEMBL8908675

CC1(C)C2CC[C@]1(C)CN(C(=O)C(c1ccccc1)C13CC4CC(CC(C4)C1)C3)C2

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 9/20 0.36
ATM Q13315 1/20 0.36
EPHX2 P34913 1/20 0.34
EPHX1 P07099 1/20 0.33
HSD11B1 P28845 1/20 0.33
ALDH1A1 P00352 2/20 0.33
DPP4 P27487 1/20 0.32
CNR2 P34972 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
P2RX7 Q99572 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908776 0.79 SIGMAR1 (0.41) SIGMAR1EPHX2EPHX1ALDH1A1
SCHEMBL8909879 0.69 SIGMAR1 (0.43) SIGMAR1HSD11B1CNR2
SCHEMBL8908667 0.69 SIGMAR1 (0.40) SIGMAR1HSD11B1ALDH1A1
SCHEMBL8910607 0.69 BPTF (0.49) SIGMAR1EPHX1HSD11B1ALDH1A1TSHR
SCHEMBL8910246 0.67 SIGMAR1 (0.43) SIGMAR1EPHX1HSD11B1TSHR
SCHEMBL8909808 0.66 SIGMAR1 (0.53) SIGMAR1HSD11B1
SCHEMBL3813465 0.65 HDAC1 (0.46) EPHX2ALDH1A1MEN1KMT2ATSHR
SCHEMBL4608058 0.65 HDAC2 (0.36) SIGMAR1EPHX2ALDH1A1TSHR
SCHEMBL3812022 0.64 HDAC1 (0.46) ATMALDH1A1MEN1KMT2ATSHR
SCHEMBL8910605 0.63 SIGMAR1 (0.60) SIGMAR1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5658923-A USED IN TREATING DISEASES RELATED TO SIGMA-RECEPTOR, SUCH AS SCHIZOPHRENIA ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-08-19 US disclosed