SCHEMBL8909415

SCHEMBL8909415

COC(=O)[C@H](C)N(C(=O)OC(C)(C)C)c1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.40
FPR2 P25090 1/20 0.40
SCN9A Q15858 1/20 0.40
TSHR P16473 1/20 0.37
MEN1 O00255 4/20 0.37
GAA P10253 1/20 0.36
KCNQ4 P56696 3/20 0.35
KCNQ5 Q9NR82 3/20 0.35
HTT P42858 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
PLA2G1B P04054 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
NOTUM Q6P988 1/20 0.35
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
LMNA P02545 1/20 0.35
CA12 O43570 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6294115 0.86 SLC6A3 (0.39) KMT2AFPR2SCN9AMEN1HTT
SCHEMBL7479568 0.86 MT-CO2 (0.46) KMT2AMEN1GAAHTTNPSR1
SCHEMBL27824592 0.86 HTT (0.35) KMT2AMEN1GAAHTTNPSR1
SCHEMBL7479440 0.86 MT-CO2 (0.46) KMT2AMEN1GAAHTTNPSR1
SCHEMBL5846260 0.86 KMT2A (0.40) KMT2AMEN1KCNQ4KCNQ5HTT
SCHEMBL8380101 0.86 KMT2A (0.45) KMT2AMEN1HTTNPSR1PLA2G1B
SCHEMBL12813777 0.84 ADRB2 (0.39) KMT2AFPR2SCN9AMEN1HTT
SCHEMBL7308442 0.84 KMT2A (0.41) KMT2AMEN1GAAHTTNPSR1
SCHEMBL2861381 0.84 XBP1 (0.37) KMT2AMEN1HTTNPSR1PLA2G1B
SCHEMBL7446003 0.84 KMT2A (0.41) KMT2AMEN1GAAHTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed
EP-0416373-A2 Amino acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-03-13 EP disclosed