SCHEMBL8909568

SCHEMBL8909568

NCCCCC(N)c1ccnc2cc(C(F)(F)F)ccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.41
NCF1 P14598 1/20 0.41
SYK P43405 1/20 0.40
PARP1 P09874 1/20 0.38
AAK1 Q2M2I8 3/20 0.38
GAK O14976 1/20 0.37
GRM4 Q14833 1/20 0.37
SLC7A5 Q01650 5/20 0.36
FERMT2 Q96AC1 1/20 0.36
PRKD3 O94806 2/20 0.36
MAP4K4 O95819 2/20 0.36
KDR P35968 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
AURKB Q96GD4 2/20 0.36
PRKD2 Q9BZL6 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
PLK4 O00444 1/20 0.36
DYRK3 O43781 1/20 0.36
CHEK2 O96017 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16013596 0.92 ADRB2 (0.44) ADRB2NCF1SYKPARP1AAK1
SCHEMBL29707948 0.85 ADRB2 (0.45) ADRB2NCF1PARP1AAK1GAK
SCHEMBL3524941 0.85 ADRB2 (0.45) ADRB2NCF1PARP1AAK1GAK
SCHEMBL4367045 0.80 FERMT2 (0.56) FERMT2
SCHEMBL28529691 0.79 ADRB2 (0.40) ADRB2NCF1SYKPARP1AAK1
SCHEMBL8907641 0.76 LOXL2 (0.49) NCF1SYKFERMT2
SCHEMBL902310 0.76 FERMT2 (0.56) FERMT2
SCHEMBL15924893 0.75 LOXL2 (0.47) NCF1SYKFERMT2
SCHEMBL5018907 0.75 ADRB2 (0.48) ADRB2NCF1PARP1AAK1GAK
SCHEMBL5548218 0.74 CCNC (0.45) ADRB2NCF1AAK1GAKGRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997048705-A1 POTASSIUM CHANNEL BLOCKERS UNIVERSITY COLLEGE LONDON (GB) 1997-12-24 WO disclosed