SCHEMBL8909812

SCHEMBL8909812

CC(O)COc1cccc(C(N)=O)c1N1CC=C(c2ccc(F)cc2)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.49
THPO P40225 1/20 0.49
LMNA P02545 1/20 0.48
PMP22 Q01453 1/20 0.48
AOC3 Q16853 2/20 0.42
ABCB1 P08183 4/20 0.41
SIGMAR1 Q99720 5/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909829 0.85 CYP2D6 (0.48) CYP2D6THPOLMNAPMP22AOC3
SCHEMBL7861690 0.77 CYP2D6 (0.71) CYP2D6THPOLMNAPMP22ABCB1
SCHEMBL19944416 0.71 DRD2 (0.61) CYP2D6THPOLMNAPMP22SIGMAR1
SCHEMBL30151910 0.69 HTT (0.65) LMNAABCB1MEN1KMT2AMAPT
SCHEMBL19944378 0.69 SIGMAR1 (0.49) CYP2D6THPOLMNAPMP22SIGMAR1
SCHEMBL7860449 0.69 CYP2D6 (0.67) CYP2D6THPOLMNAPMP22ABCB1
SCHEMBL19944866 0.69 PARP1 (0.47) CYP2D6THPOLMNAPMP22SIGMAR1
SCHEMBL6021254 0.66 CYP2D6 (1.00) CYP2D6THPOLMNAPMP22ABCB1
Hydrochloric Acid SCHEMBL2001258 0.65 LMNA (1.00) CYP2D6THPOLMNAPMP22ABCB1
SCHEMBL7862476 0.63 ABCB1 (0.65) LMNAABCB1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5698565-A TREATMENT OF PSYCHOTIC DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-12-16 US claimed