SCHEMBL8911633

SCHEMBL8911633

C=C1c2ccccc2N(C)C1(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.41
ALDH1A1 P00352 4/20 0.41
GAA P10253 3/20 0.41
MCL1 Q07820 2/20 0.41
PAX8 Q06710 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 4/20 0.35
MAPT P10636 4/20 0.35
HPGD P15428 2/20 0.35
CES1 P23141 2/20 0.35
TTR P02766 1/20 0.35
NSD2 O96028 1/20 0.35
APP P05067 1/20 0.35
SNCA P37840 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HTT P42858 2/20 0.34
MAPK1 P28482 1/20 0.34
CACNA1B Q00975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23520298 0.77 ALDH1A1 (0.36) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL17275723 0.75 ALDH1A1 (0.50) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL26327450 0.75 KMT2A (0.42) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL25682366 0.73 GAA (0.48) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL28060229 0.71 GAA (0.37) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL10345602 0.66 NR1H3 (0.35) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL15907068 0.65 ALDH1A1 (0.39) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL2393621 0.65 LMNA (0.57) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL29565250 0.64 ALDH1A1 (0.47) LMNAALDH1A1GAAMCL1PAX8
SCHEMBL21726115 0.64 MAPT (0.40) LMNAALDH1A1GAAMCL1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3087094-B1 BETA-HAIRPIN PEPTIDOMIMETICS AS SELECTIVE ELASTASE INHIBITORS POLYPHOR AG (CH) 2022-06-01 EP disclosed
EP-0489655-B1 Indolino-spiro-benzoxazine photochromic compounds and process for their preparation ESSILOR INT (FR) 1997-05-28 EP disclosed
EP-0402228-B1 Indolino-spiro-oxazine photochromic compounds having a five-membered ring, process for their preparation and photochromic compositions and materials containing them ESSILOR INT (FR) 1996-01-03 EP disclosed
EP-0407237-B1 Indolino-spiro-oxazine photochromic compounds, process for their preparation and photochromic compositions and materials containing them ESSILOR INT (FR) 1995-11-29 EP disclosed
US-5233038-A PHOTOCHRONIC COMPOUNDS OF THE INDOLINO-SPIRO-BENZOXAZINE TYPE ESSILOR INTERNATIONAL (COMPAGNIE GENERALE D'OPTIQUE) (FR) 1993-08-03 US disclosed
EP-0489655-A1 Indoline-spiro-benzoxazine photochromic compounds and process for their preparation ESSILOR INTERNATIONAL Compagnie Générale d'Optique (FR) 1992-06-10 EP disclosed
EP-0407237-A2 Indolino-spiro-oxazine photochromic compounds, process for their preparation and photochromic compositions and materials containing them ESSILOR INTERNATIONAL (Compagnie Générale d'Optique) (FR) 1991-01-09 EP disclosed
EP-0402228-A2 Indolino-spiro-oxazine photochromic compounds having a five-membered ring, process for their preparation and photochromic compositions and materials containing them ESSILOR INTERNATIONAL (Compagnie Générale d'Optique) (FR) 1990-12-12 EP disclosed
US-4542224-A Process for preparing cationic methine dyestuffs BAYER AKTIENGESELLSCHAFT (DE) 1985-09-17 US disclosed
EP-0092698-B1 PROCESS FOR THE PREPARATION OF CATIONIC METHINE DYES BAYER AG (DE) 1985-06-26 EP disclosed
EP-0092698-A1 Process for the preparation of cationic methine dyes BAYER AG (DE) 1983-11-02 EP disclosed