SCHEMBL8912501

SCHEMBL8912501

O=C(O)n1c(C2CCCCC2)cc(=O)c2cc(F)c(O)c(F)c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.34
NR1I2 O75469 1/20 0.33
KDM4B O94953 1/20 0.33
CHRM1 P11229 1/20 0.33
TBXA2R P21731 1/20 0.33
ADRA1A P35348 1/20 0.33
DOHH Q9BU89 1/20 0.33
KDM4E B2RXH2 2/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
CYP1A2 P05177 1/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HIF1A Q16665 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7121568 0.74 TOP2A (0.41) EGLN1KDM4EMEN1KMT2ALMNA
SCHEMBL7123595 0.62 ALDH1A1 (0.41) KDM4EMAPTKMT2AMAPK1SMN1; SMN2
SCHEMBL15971194 0.60 CNR2 (0.41) KDM4EMEN1KMT2ACYP1A2SMN1; SMN2
SCHEMBL21632762 0.59 ACMSD (0.41) KDM4EMEN1MAPTKMT2ASMN1; SMN2
SCHEMBL11756192 0.59 KDM4E (0.50) KDM4EMEN1MAPTKMT2APTGDR2
Bicarbonate SCHEMBL9629020 0.59 KMO (0.46) KDM4EKMT2APTGDR2SMN1; SMN2HIF1A
SCHEMBL8096676 0.58 TOP2A (0.47) CHRM1KDM4EMAPTLMNACYP1A2
SCHEMBL11374138 0.56 KDM4E (0.50) KDM4EMEN1MAPTKMT2APTGDR2
SCHEMBL9787018 0.55 KDM4E (0.45) NR1I2KDM4BCHRM1TBXA2RADRA1A
SCHEMBL11335917 0.54 KDM4E (0.44) EGLN1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0793656-A1 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1997-09-10 EP disclosed
WO-1996016046-A2 NOVEL BENZYL PYRIMIDINES F. HOFFMANN-LA ROCHE AG (CH) 1996-05-30 WO disclosed