SCHEMBL8912823

SCHEMBL8912823

C[N+]1([O-])CCC2(CC1)Cc1ccc(NS(C)(=O)=O)cc1CO2

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.34
PGR P06401 1/20 0.34
NR3C2 P08235 1/20 0.34
AR P10275 1/20 0.34
CYP2C9 P11712 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
TDP2 O95551 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912474 0.81 ADRA1D (0.41)
Hydrochloric Acid SCHEMBL8912790 0.81 HTR6 (0.37) NR3C1PGRNR3C2ARTDP2
Hydrochloric Acid SCHEMBL8913394 0.73 KCNH2 (0.50)
Hydrochloric Acid SCHEMBL8570970 0.69 KDM4E (0.43)
Hydrochloric Acid SCHEMBL8922961 0.68 KCNH2 (0.43)
SCHEMBL24388772 0.67 BRD4 (0.43) NR3C2CA12CA1CA2CA9
SCHEMBL24388853 0.66 BRPF1 (0.43) CYP2C9
SCHEMBL24389272 0.65 ALDH1A1 (0.41) NR3C2CA12CA1CA2CA9
SCHEMBL8913770 0.64 ADRA1D (0.41)
Hydrochloric Acid SCHEMBL8914251 0.64 HTR6 (0.38) NR3C1PGRNR3C2ARCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed