SCHEMBL8912474

SCHEMBL8912474

CN1CCC2(CC1)Cc1ccc(NS(C)(=O)=O)cc1CO2

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 4/20 0.41
ADRA1A P35348 3/20 0.41
ADRA1B P35368 2/20 0.40
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8913394 0.85 KCNH2 (0.50) ADRA1DADRA1AADRA1BKCNH2
Hydrochloric Acid SCHEMBL8912790 0.84 HTR6 (0.37)
SCHEMBL8912823 0.81 NR3C1 (0.34)
SCHEMBL24388853 0.80 BRPF1 (0.43)
Hydrochloric Acid SCHEMBL8570970 0.78 KDM4E (0.43) ADRA1DADRA1AKCNH2
Hydrochloric Acid SCHEMBL8922961 0.77 KCNH2 (0.43) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL8564005 0.73 ADRA1D (0.66) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL8913639 0.72 ADRA1D (0.46) ADRA1DADRA1AADRA1BKCNH2
SCHEMBL24388772 0.70 BRD4 (0.43)
SCHEMBL24389272 0.67 ALDH1A1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed