SCHEMBL8914593

SCHEMBL8914593

O=[N+]([O-])c1ccc2c(c1)SC1(CCNCC1)S2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
MAPT P10636 1/20 0.47
RAB9A P51151 1/20 0.47
SNCA P37840 4/20 0.42
ADRA2A P08913 1/20 0.41
PNMT P11086 1/20 0.41
ADRB1 P08588 1/20 0.40
SIRT6 Q8N6T7 1/20 0.40
NOX1 Q9Y5S8 1/20 0.39
CYP3A4 P08684 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
SLC6A4 P31645 1/20 0.37
CYP2C19 P33261 1/20 0.37
THPO P40225 1/20 0.37
HTR3A P46098 1/20 0.37
HTR3D Q70Z44 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912806 0.72 KCNJ1 (0.60) KCNJ1KCNH2
SCHEMBL8913631 0.72 TDP1 (0.51) NPC1MAPTRAB9ATDP1ALDH1A1
SCHEMBL12862872 0.70 ADRA2A (0.41) MAPTSNCAADRA2APNMTADRB1
SCHEMBL1144860 0.67 SNCA (0.56) SNCANOX1CYP3A4TDP1ALDH1A1
SCHEMBL9698085 0.67 SNCA (0.56) SNCANOX1CYP3A4TDP1ALDH1A1
SCHEMBL8469291 0.66 SNCA (0.51) NPC1MAPTRAB9ASNCANOX1
SCHEMBL11918666 0.65 PNMT (0.43) MAPTADRA2APNMTADRB1SIRT6
SCHEMBL1208092 0.65 SNCA (0.84) NPC1MAPTRAB9ASNCANOX1
SCHEMBL29625234 0.65 SNCA (0.84) NPC1MAPTRAB9ASNCANOX1
SCHEMBL3031049 0.65 SNCA (0.68) NPC1MAPTRAB9ASNCANOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed