SCHEMBL8916189

SCHEMBL8916189

COc1ccc2c(ccc3c(C(N)=O)nn(-c4ccc(S(N)(=O)=O)cc4)c32)c1Cl

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.52
PTGS1 P23219 6/20 0.52
CA1 P00915 6/20 0.44
CA2 P00918 6/20 0.44
CA9 Q16790 5/20 0.44
CA4 P22748 4/20 0.44
SMN1; SMN2 Q16637 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9234798 0.92 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA9
SCHEMBL8917392 0.92 PTGS2 (0.57) PTGS2PTGS1CA1CA2CA9
SCHEMBL8916244 0.92 PTGS2 (0.42) PTGS2PTGS1
SCHEMBL8917741 0.88 CA9 (0.52) PTGS2PTGS1CA1CA2CA9
SCHEMBL9229223 0.82 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8917527 0.82 PTGS2 (0.45) PTGS2PTGS1SMN1; SMN2
SCHEMBL9235122 0.81 PTGS2 (0.54) PTGS2PTGS1
SCHEMBL9233583 0.81 PTGS2 (0.52) PTGS2PTGS1CA1CA2CA9
SCHEMBL8920714 0.78 PTGS2 (0.46) PTGS2CA1CA2CA9CA4
SCHEMBL9231677 0.77 CA1 (0.58) PTGS2PTGS1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996009293-A1 BENZ[g]INDAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO claimed
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed
WO-1996010015-A1 CRYPTOLEPINE ANALOGS WITH HYPOGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1996-04-04 WO disclosed
WO-1996009293-A1 BENZ[g]INDAZOLYL DERIVATIVES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-03-28 WO disclosed