SCHEMBL8920714

SCHEMBL8920714

CCOC(=O)c1nn(-c2ccc(S(C)(=O)=O)cc2)c2c1ccc1c(Cl)c(OC)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.46
NPBWR1 P48145 1/20 0.43
MAPT P10636 4/20 0.42
CA9 Q16790 4/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA4 P22748 3/20 0.42
APP P05067 2/20 0.42
CASP1 P29466 1/20 0.42
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 2/20 0.41
ADORA1 P30542 2/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP6 P55212 1/20 0.41
HSD17B10 Q99714 1/20 0.41
CA12 O43570 1/20 0.41
CHRNA7 P36544 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917527 0.92 PTGS2 (0.45) PTGS2NPBWR1MAPTALDH1A1L3MBTL1
SCHEMBL8917741 0.91 CA9 (0.52) PTGS2MAPTCA9CA1CA2
SCHEMBL9229223 0.88 PTGS2 (0.40) PTGS2MAPTADORA1
SCHEMBL8916244 0.87 PTGS2 (0.42) PTGS2
SCHEMBL8917392 0.82 PTGS2 (0.57) PTGS2CA9CA1CA2CA4
SCHEMBL8916189 0.78 PTGS2 (0.52) PTGS2CA9CA1CA2CA4
SCHEMBL9234798 0.78 PTGS2 (0.52) PTGS2CA9CA1CA2CA4
SCHEMBL8918689 0.77 PTGS2 (0.51) PTGS2
SCHEMBL8918668 0.73 CA12 (0.46) PTGS2CA9CA1CA2ALDH1A1
SCHEMBL8917550 0.72 PTGS2 (0.40) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696143-A ARTHRITIS THERAPY G.D. SEARLE & CO. 1997-12-09 US disclosed