SCHEMBL8917035

SCHEMBL8917035

CCc1c(CCN2CCC(c3cc4ccccc4o3)CC2)sc2c1CCN(C(C)=O)C2

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 8/20 0.46
BCHE P06276 5/20 0.43
MCHR1 Q99705 2/20 0.38
TP53 P04637 6/20 0.38
MAPT P10636 6/20 0.38
OXTR P30559 1/20 0.38
GAA P10253 1/20 0.36
POLB P06746 1/20 0.36
HTR3A P46098 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917865 0.90 MAPT (0.38) ACHEBCHEMCHR1TP53MAPT
Hydrochloric Acid SCHEMBL8918152 0.87 ACHE (0.39) ACHEBCHEMCHR1TP53MAPT
SCHEMBL8917705 0.85 DRD2 (0.52) MCHR1TP53MAPTGAAPOLB
SCHEMBL8919111 0.83 DRD2 (0.51)
Hydrochloric Acid SCHEMBL8917305 0.83 ACHE (0.36) ACHEBCHEMCHR1TP53MAPT
SCHEMBL8916565 0.81 MAOA (0.41) MCHR1TP53MAPTPOLBKDM4E
SCHEMBL8916433 0.80 TP53 (0.40) MCHR1TP53MAPTGAAPOLB
Oxalic Acid SCHEMBL8916497 0.80 DRD2 (0.45)
SCHEMBL8916426 0.79 MAPT (0.40) MCHR1TP53MAPTGAAPOLB
SCHEMBL8916930 0.78 SLC6A4 (0.52) MCHR1TP53MAPTGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed