SCHEMBL8917174

SCHEMBL8917174

CC(C)(C)OC(=O)c1ncc(N)c(N2CCNCC2)n1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.38
HRH3 Q9Y5N1 3/20 0.36
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
CSNK1A1 P48729 1/20 0.34
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
KCNH2 Q12809 1/20 0.33
PIM1 P11309 1/20 0.33
PIM3 Q86V86 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917059 0.81 PRKD1 (0.36) HRH4HRH3ALDH1A1KDM4ECSNK1A1
SCHEMBL30384988 0.81 CRBN (0.38) HRH4HRH3CYP2D6TSHRCLK4
SCHEMBL28605663 0.81 CRBN (0.38) HRH4HRH3CYP2D6TSHRCLK4
SCHEMBL14854851 0.74 ALDH1A1 (0.34) ALDH1A1KDM4EHPGD
SCHEMBL8915788 0.74 HTR2C (0.40) HRH3
SCHEMBL5502924 0.74 KDM4E (0.52) ALDH1A1KDM4ESMN1; SMN2CYP2D6TSHR
SCHEMBL5502137 0.70 NCF1 (0.49) ALDH1A1KDM4ECYP2D6TSHRCLK4
SCHEMBL15415762 0.69 ALDH1A1 (0.35) ALDH1A1KDM4ECSNK1A1CYP2D6TSHR
SCHEMBL27591250 0.68 KDM4E (0.56) ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL20423547 0.68 CRBN (0.57) ALDH1A1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686610-A Pyridyl piperazine compound PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed