SCHEMBL5502137

SCHEMBL5502137

COc1ccc2nc(C(=O)OC(C)(C)C)nc(N3CCNCC3)c2c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.49
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
TP53 P04637 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
PDE10A Q9Y233 1/20 0.45
USP2 O75604 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ILK Q13418 1/20 0.43
MTNR1B P49286 2/20 0.42
NTSR1 P30989 2/20 0.42
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR3A P46098 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502924 0.84 KDM4E (0.52) NCF1CYP1A2CYP3A4TP53CYP2D6
SCHEMBL5502143 0.82 NCF1 (0.50) NCF1CYP1A2CYP3A4TP53CYP2D6
SCHEMBL16416202 0.72 HTR6 (0.63) NCF1CYP1A2CYP3A4TP53CYP2D6
SCHEMBL3679159 0.71 HTR1A (0.53) NCF1CYP1A2CYP3A4TP53CYP2D6
SCHEMBL1222766 0.71 CYP1A2 (0.76) NCF1CYP1A2CYP3A4CYP2D6TSHR
SCHEMBL16416324 0.71 SLC2A1 (0.54) KMT2AMEN1KDM4EMTNR1BHTR6
SCHEMBL8917174 0.70 HRH4 (0.38) CYP2D6TSHRCLK4KDM4EALDH1A1
SCHEMBL4190466 0.69 NCF1 (0.56) NCF1KMT2AMEN1KDM4EHTR3E
Trifluoroacetic Acid SCHEMBL30619102 0.69 NCF1 (0.50) NCF1CYP1A2CYP3A4TP53CYP2D6
SCHEMBL2708405 0.69 ADRB2 (0.72) NCF1CYP1A2CYP3A4TP53CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218353-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA UK LTD (GB) 2007-10-17 EP disclosed
EP-1272185-B1 USE OF QUINAZOLINE DERIVATIVES AS ANGIOGENESIS INHIBITORS ASTRAZENECA AB (SE) 2005-07-27 EP disclosed