SCHEMBL8917192

SCHEMBL8917192

CCOC(=O)c1c(C)nc(N)c(C#N)c1-c1ccc(Cl)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.65
KDM4E B2RXH2 7/20 0.65
HPGD P15428 3/20 0.65
LMNA P02545 4/20 0.61
KMT2A Q03164 3/20 0.61
L3MBTL1 Q9Y468 1/20 0.58
MEN1 O00255 2/20 0.57
RECQL P46063 1/20 0.57
HIF1A Q16665 1/20 0.57
CACNB4 O00305 2/20 0.53
CACNA1A O00555 2/20 0.53
CACNA1G O43497 2/20 0.53
CACNG3 O60359 2/20 0.53
CACNA1F O60840 2/20 0.53
CACNA1H O95180 2/20 0.53
ACHE P22303 2/20 0.53
CACNB3 P54284 2/20 0.53
CACNA2D1 P54289 2/20 0.53
CACNG7 P62955 2/20 0.53
CACNA1B Q00975 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918577 0.89 ALDH1A1 (0.72) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL8918613 0.89 GAA (0.68) ALDH1A1KDM4EHPGDKMT2AL3MBTL1
SCHEMBL8917637 0.86 CACNB4 (0.54) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL6137355 0.80 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL6137213 0.78 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL22573316 0.77 KDM4E (0.76) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL6137173 0.75 AR (0.57) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL32688181 0.75 ALDH1A1 (0.65) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL31442597 0.74 SMN1; SMN2 (0.81) ALDH1A1KDM4EHPGDLMNAKMT2A
SCHEMBL8975579 0.74 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670525-A Substituted 4-phenyl-6-amino-nicotinic acid compounds useful in the treatment of CNS disorders BAYER AKTIENGESELLSCHAFT (DE) 1997-09-23 US claimed
EP-0705820-A1 6-Amino-nicotinic acid derivatives and their use as selective K-channel modulators BAYER AG (DE) 1996-04-10 EP claimed
US-5670525-A Substituted 4-phenyl-6-amino-nicotinic acid compounds useful in the treatment of CNS disorders BAYER AKTIENGESELLSCHAFT (DE) 1997-09-23 US disclosed
EP-0705820-A1 6-Amino-nicotinic acid derivatives and their use as selective K-channel modulators BAYER AG (DE) 1996-04-10 EP disclosed