SCHEMBL8975579

SCHEMBL8975579

COc1ccc(-c2c(C#N)c(N)nc(C)c2C(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
MAPT P10636 6/20 0.55
NPSR1 Q6W5P4 5/20 0.55
KDM4E B2RXH2 5/20 0.55
RXFP1 Q9HBX9 3/20 0.55
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
HPGD P15428 1/20 0.53
MAPK1 P28482 1/20 0.53
GAA P10253 3/20 0.53
ADORA1 P30542 5/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ADORA2A P29274 2/20 0.50
ADRA2A P08913 1/20 0.50
HTT P42858 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ELAVL1 Q15717 1/20 0.48
POLB P06746 1/20 0.47
FNTA P49354 1/20 0.46
FNTB P49356 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918613 0.86 GAA (0.68) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL8974906 0.86 HSD17B10 (0.68) ALDH1A1KDM4ERXFP1HPGDADORA1
SCHEMBL8975128 0.81 HTT (0.48) ALDH1A1MAPTKDM4ERXFP1MEN1
SCHEMBL8918577 0.75 ALDH1A1 (0.72) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL3359383 0.74 KDM4E (0.60) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL8917192 0.74 ALDH1A1 (0.65) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL17747485 0.73 ALDH1A1 (0.76) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL15286708 0.73 ADORA1 (0.50) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL13914641 0.73 ALDH1A1 (0.74) ALDH1A1MAPTNPSR1KDM4ERXFP1
SCHEMBL13913746 0.72 ADORA1 (0.80) ALDH1A1MAPTNPSR1KDM4ERXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705820-A1 6-Amino-nicotinic acid derivatives and their use as selective K-channel modulators BAYER AG (DE) 1996-04-10 EP disclosed