SCHEMBL8919989

SCHEMBL8919989

O=C(O)N[C@@H](CCC[C@H](O)CCl)Cc1ccc2ccccc2c1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.41
MME P08473 5/20 0.41
ACE P12821 5/20 0.41
CPA1 P15085 2/20 0.41
ACE2 Q9BYF1 2/20 0.41
CYP1A2 P05177 1/20 0.40
FCER2 P06734 2/20 0.40
TACR1 P25103 1/20 0.39
MMP9 P14780 2/20 0.39
MMP8 P22894 2/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
CA2 P00918 1/20 0.39
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918697 0.76 TACR1 (0.46) MMEACECPA1ACE2CYP1A2
SCHEMBL8918692 0.76 TACR1 (0.46) MMEACECPA1ACE2CYP1A2
SCHEMBL7291165 0.75 HTR2A (0.39) CYP1A2FCER2MMP9HDAC1HDAC8
SCHEMBL8919990 0.74 HTR2A (0.46) PIN1MMEACECPA1ACE2
SCHEMBL8921872 0.72 CTSG (0.52) PIN1MMEACECPA1ACE2
SCHEMBL8921880 0.72 CTSG (0.52) PIN1MMEACECPA1ACE2
SCHEMBL21628079 0.71 MME (0.50) MMECYP1A2
SCHEMBL8919979 0.71 MME (0.47) MMEACECPA1ACE2FCER2
SCHEMBL8919984 0.71 MME (0.44) MMEACECPA1ACE2FCER2
SCHEMBL10961713 0.70 MMP9 (0.51) MMEACECPA1ACE2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed