SCHEMBL8921880

SCHEMBL8921880

O=C(O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)CCl

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSG P08311 2/20 0.52
CMA1 P23946 2/20 0.52
MME P08473 4/20 0.51
ACE P12821 4/20 0.51
CPA1 P15085 2/20 0.51
ACE2 Q9BYF1 2/20 0.51
TACR1 P25103 1/20 0.49
MMP9 P14780 2/20 0.49
MMP8 P22894 2/20 0.49
CA2 P00918 1/20 0.48
CTSB P07858 3/20 0.46
CTSS P25774 3/20 0.46
CTSL P07711 2/20 0.46
CTSK P43235 2/20 0.46
FCER2 P06734 2/20 0.46
PIN1 Q13526 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8921872 1.00 CTSG (0.52) CTSGCMA1MMEACECPA1
SCHEMBL3628827 0.86 MME (0.56) MMEACECPA1ACE2TACR1
SCHEMBL4291672 0.84 CTSG (0.65) CTSGCMA1MMEACE
SCHEMBL6942656 0.84 CTSG (0.65) CTSGCMA1MMEACE
SCHEMBL5664274 0.84 CTSG (0.65) CTSGCMA1MMEACE
SCHEMBL2345995 0.80 MMP9 (0.47) MMEACECPA1ACE2TACR1
SCHEMBL2343629 0.80 MME (0.50) MMEACECPA1ACE2TACR1
SCHEMBL8201136 0.78 FCER2 (0.69) MMEACECPA1ACE2MMP9
SCHEMBL8201134 0.78 FCER2 (0.69) MMEACECPA1ACE2MMP9
SCHEMBL8918692 0.77 TACR1 (0.46) MMEACECPA1ACE2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652369-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1997-07-29 US disclosed
US-5554756-A PROTEASE INHIBITOR HOFFMANN-LA ROCHE INC. (US) 1996-09-10 US disclosed
US-5446161-A Protease inhibitor, viricides HOFFMANN-LA ROCHE INC. (US) 1995-08-29 US disclosed