SCHEMBL9542930

SCHEMBL9542930

NC(=O)CN1C(=O)C(N)CC(c2ccc(Cl)c(Cl)c2)c2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.45
SLC6A4 P31645 11/20 0.45
SLC6A3 Q01959 11/20 0.45
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922239 0.89 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3CYP2D6CYP2C19
SCHEMBL9540219 0.88 CCKBR (0.47) CYP2C19
SCHEMBL9541670 0.87 CCKBR (0.51) CYP2C19
SCHEMBL8919676 0.85 CCKBR (0.57) SLC6A2SLC6A4SLC6A3
SCHEMBL8920848 0.85 CYP2C19 (0.47) CYP2C19
SCHEMBL9540184 0.84 CYP2C19 (0.43) CYP2C19
SCHEMBL9541664 0.84 CCKBR (0.48) CYP2C19
SCHEMBL9544115 0.80 CYP2C19 (0.46) CYP2C19
SCHEMBL9542926 0.80 CCKBR (0.49) CYP2C19
SCHEMBL9541282 0.78 CCKBR (0.69)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed