SCHEMBL9540219

SCHEMBL9540219

NC(=O)CN1C(=O)C(N)CC(c2ccc(Cl)cc2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 12/20 0.47
CYP2C19 P33261 1/20 0.43
GPBAR1 Q8TDU6 1/20 0.37
PDPK1 O15530 1/20 0.37
PYGL P06737 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8920848 0.91 CYP2C19 (0.47) CCKBRCYP2C19
SCHEMBL9540184 0.89 CYP2C19 (0.43) CCKBRCYP2C19
SCHEMBL9541664 0.89 CCKBR (0.48) CCKBRCYP2C19
SCHEMBL8923711 0.89 CCKBR (0.47) CCKBRCYP2C19PDPK1
SCHEMBL9541670 0.88 CCKBR (0.51) CCKBRCYP2C19
SCHEMBL9542930 0.88 SLC6A2 (0.45) CYP2C19
SCHEMBL9542926 0.87 CCKBR (0.49) CCKBRCYP2C19
SCHEMBL8919215 0.84 CCKBR (0.67) CCKBR
SCHEMBL9544115 0.82 CYP2C19 (0.46) CYP2C19
SCHEMBL9366810 0.79 CYP2C19 (0.47) CCKBRCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed