SCHEMBL8922129

SCHEMBL8922129

Cc1cccc(N(C(N)=O)C2CCCC(c3ccccc3)N(CN(C=O)C34CC5CC(CC(C5)C3)C4)C2=O)c1

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
MAPT P10636 2/20 0.32
ALOX15 P16050 1/20 0.32
PKM P14618 1/20 0.32
RAB9A P51151 2/20 0.32
GAA P10253 1/20 0.32
LMNA P02545 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
UTS2R Q9UKP6 1/20 0.32
CCKBR P32239 3/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9362231 0.86 ALDH1A1 (0.34) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL8922451 0.85 LMNA (0.38) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL8922740 0.84 HSD11B1 (0.33) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL8922121 0.81 ALDH1A1 (0.39) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL9366881 0.78 ALDH1A1 (0.34) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL8920349 0.77 RAMP1 (0.42) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL9541317 0.74 LMNA (0.38) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL8921847 0.71 LMNA (0.34) RAB9ALMNASMN1; SMN2
SCHEMBL8926039 0.71 DRD2 (0.32) ALDH1A1MAPTALOX15PKMRAB9A
SCHEMBL9365841 0.69 NPSR1 (0.32) ALDH1A1MAPTALOX15PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643904-A Substituted hexahdryoazepinones and tetrahydrobenzazepinones PFIZER INC. (US) 1997-07-01 US disclosed
US-5484917-A FOR TREATMENT AND PREVENTION OF GASTROINTESTINAL DISORDERS, PAIN AND ANXIETY PFIZER INC. (US) 1996-01-16 US disclosed
WO-1993015059-A1 3-PHENYLUREIDO-AZEPIN-2-ONES AND -BENZAZEPIN-2-ONES USEFUL AS CHOLECYSTOKININ ANTAGONISTS PFIZER INC. (US) 1993-08-05 WO disclosed