SCHEMBL8923587

SCHEMBL8923587

N#CC(CSP(=O)(O)O)Cc1ccc(Cl)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GGPS1 O95749 1/20 0.43
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
MAPK1 P28482 1/20 0.37
CYP2C19 P33261 1/20 0.37
IDO1 P14902 5/20 0.37
DPP4 P27487 3/20 0.36
HDAC8 Q9BY41 5/20 0.36
FAP Q12884 2/20 0.35
DPP8 Q6V1X1 2/20 0.35
DPP9 Q86TI2 2/20 0.35
DPP7 Q9UHL4 2/20 0.35
EPHX1 P07099 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HTT P42858 2/20 0.35
CA1 P00915 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8922306 0.81 CTSC (0.41) CYP1A2CYP2C19DPP4FAPDPP8
SCHEMBL8925358 0.76 GGPS1 (0.39) GGPS1HTTCA1CA14
SCHEMBL8921479 0.72 LAP3 (0.44) CYP1A2
SCHEMBL11350035 0.71 GAA (0.42) CYP1A2CYP3A4CYP2C9CYP2C19DPP4
SCHEMBL4657319 0.70 IDO1 (0.48) GGPS1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL3762617 0.67 IDO1 (0.46) CYP1A2CYP3A4CYP2C9MAPK1CYP2C19
SCHEMBL21056096 0.67 IDO1 (0.46) CYP1A2CYP3A4CYP2C9MAPK1CYP2C19
SCHEMBL11858796 0.66 MEN1 (0.49) CYP1A2CYP2C19IDO1HTT
SCHEMBL24191243 0.65 CYP1A2 (0.55) GGPS1CYP1A2CYP3A4CYP2C9MAPK1
SCHEMBL11861718 0.65 ALDH1A1 (0.43) GGPS1CYP1A2CYP3A4CYP2C9MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5210264-A S-(2,4-dichlorobenzyl)-β-cyanoethyl phosphorothioate diester ISIS PHARMACEUTICALS, INC. (US) 1993-05-11 US claimed
US-5644048-A Process for preparing phosphorothioate oligonucleotides ISIS PHARMACEUTICALS, INC. (US) 1997-07-01 US disclosed
WO-1994019363-A1 PROCESS FOR PREPARING PHOSPHOROTHIOATE OLIGONUCLEOTIDES ISIS PHARMACEUTICALS, INC. (US) 1994-09-01 WO disclosed
US-5210264-A S-(2,4-dichlorobenzyl)-β-cyanoethyl phosphorothioate diester ISIS PHARMACEUTICALS, INC. (US) 1993-05-11 US disclosed
US-5210264-A S-(2,4-dichlorobenzyl)-β-cyanoethyl phosphorothioate diester ISIS PHARMACEUTICALS, INC. (US) 1993-05-11 US disclosed
US-5210264-A S-(2,4-dichlorobenzyl)-β-cyanoethyl phosphorothioate diester ISIS PHARMACEUTICALS, INC. (US) 1993-05-11 US disclosed