SCHEMBL8924717

SCHEMBL8924717

COc1c(C)c(C)c(OC(C)C)c(C)c1CN(C)C(COc1cc(C)ccc1C(C)C)OS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
ALDH1A1 P00352 6/20 0.35
KDM4E B2RXH2 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 1/20 0.35
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GALR3 O60755 1/20 0.34
NR2F2 P24468 1/20 0.34
HTT P42858 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
MAPT P10636 3/20 0.33
MAPK1 P28482 1/20 0.33
ATM Q13315 1/20 0.33
ADRB2 P07550 2/20 0.32
NPBWR1 P48145 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8924712 0.78 ADRA1D (0.51) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8922600 0.75 ADRA1D (0.57) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8924115 0.69 ALDH1A1 (0.54) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8924282 0.67 ADRA1D (0.58) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8923620 0.64 ADRA1D (0.74) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8923441 0.63 KMT2A (0.56) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL25484230 0.60 ADRB2 (0.56) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL19308590 0.58 LMNA (0.50) ALDH1A1KDM4ETDP1LMNASMN1; SMN2
SCHEMBL15791678 0.57 ADRB2 (0.64) KMT2AMEN1ALDH1A1KDM4ETDP1
SCHEMBL8246277 0.57 ALDH1A1 (0.55) KMT2AMEN1ALDH1A1KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5624961-A Benzylaminoethoxybenzene derivatives, production thereof and use thereof JAPAN TOBACCO INC. (JP) 1997-04-29 US disclosed
EP-0693474-A1 NOVEL BENZYLAMINOETHOXYBENZENE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Toyo Boseki Kabushiki Kaisha (JP) 1996-01-24 EP disclosed