SCHEMBL8924801

SCHEMBL8924801

COc1ccc(NC(=O)OC(C)(C)C)c(CCCC(C)=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 6/20 0.43
MTNR1B P49286 5/20 0.43
KDM4E B2RXH2 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
MAOA P21397 1/20 0.41
SLC6A2 P23975 1/20 0.41
RAB9A P51151 1/20 0.41
SLC6A3 Q01959 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 2/20 0.39
POLB P06746 2/20 0.39
NR1I2 O75469 1/20 0.38
HPGD P15428 1/20 0.38
APOBEC3A P31941 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8502442 0.93 MAPT (0.46) MTNR1AMTNR1BKDM4ENPC1LMNA
SCHEMBL8505209 0.85 MTNR1A (0.39) MTNR1AMTNR1BKDM4ENPC1MAPT
SCHEMBL24254051 0.83 ALDH1A1 (0.46) MAPTSMN1; SMN2ALDH1A1NR1I2
SCHEMBL7963161 0.83 KMT2A (0.40) TP53CYP3A4MAPTSMN1; SMN2ALDH1A1
SCHEMBL7962276 0.79 AKR1C3 (0.41) MTNR1AMTNR1BKDM4ENPC1MAPT
SCHEMBL8762406 0.78 ALDH1A1 (0.41) KDM4ENPC1RAB9AALDH1A1NR1I2
SCHEMBL2156670 0.78 AKR1C3 (0.48) SMN1; SMN2ALDH1A1NR1I2
SCHEMBL3584387 0.78 PIK3CG (0.41) MTNR1AMTNR1BKDM4ELMNAMAPT
SCHEMBL3225589 0.77 NR1I2 (0.41) LMNAALDH1A1POLBNR1I2
SCHEMBL13316203 0.77 PIK3CG (0.46) SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684034-A INHIBITORS OF HUMAN NON-PANCREATIC SECRETORY PHOSPHOLIPASE A2, TREATMENT OF SEPTIC SHOCK, TRAUMA, RESPIRATORY DISORDERS, RHEUMATIC ARTHRITIS, INHIBITORS OF ARACHIDONIC ACID RELEASE ELI LILLY AND COMPANY (US) 1997-11-04 US disclosed