SCHEMBL8925003

SCHEMBL8925003

Cc1cc(Sc2ccccn2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.41
PTGS1 P23219 1/20 0.41
ALDH1A1 P00352 3/20 0.40
CA2 P00918 1/20 0.39
MAPT P10636 2/20 0.37
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PDE7A Q13946 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926763 0.86 SLC9A1 (0.37)
SCHEMBL8927147 0.86 CA2 (0.39) PTGS2PTGS1ALDH1A1CA2MAPT
SCHEMBL7802693 0.83 SLC9A1 (0.57)
SCHEMBL8925113 0.81 CA12 (0.45) ALDH1A1CA2HPGD
SCHEMBL8926916 0.80 PDE7A (0.41) PTGS2PTGS1PDE7A
SCHEMBL8925101 0.79 ALDH1A1 (0.37) PTGS2ALDH1A1CA2MAPTMEN1
SCHEMBL8927186 0.78 ALDH1A1 (0.40) PTGS2ALDH1A1
SCHEMBL8926776 0.78 PTGS1 (0.38) PTGS2PTGS1
SCHEMBL8926231 0.75 RHEB (0.43) ALDH1A1MAPTHPGDNPSR1
SCHEMBL8925087 0.75 PDE4B (0.41) CA2MAPTMEN1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US disclosed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN disclosed