SCHEMBL8926776

SCHEMBL8926776

Cc1cc(Sc2cccnc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
MKNK1 Q9BUB5 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
CYP11B2 P19099 1/20 0.36
TYMS P04818 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926916 0.87 PDE7A (0.41) PTGS1PTGS2
SCHEMBL8926714 0.86 PTGS1 (0.36) PTGS1PTGS2
SCHEMBL8925113 0.85 CA12 (0.45)
SCHEMBL7800443 0.84 SLC9A1 (0.56)
SCHEMBL8925087 0.81 PDE4B (0.41)
SCHEMBL8926763 0.80 SLC9A1 (0.37)
SCHEMBL8926370 0.80 SLC6A9 (0.36)
SCHEMBL8926231 0.79 RHEB (0.43)
SCHEMBL8925017 0.78 KDM4E (0.39) PTGS1PTGS2
SCHEMBL8925003 0.78 PTGS2 (0.41) PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US disclosed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN disclosed