SCHEMBL8926718

SCHEMBL8926718

CCc1cc(Sc2ccc(F)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AGBL2 Q5U5Z8 1/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
PTGS2 P35354 4/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
PTGS1 P23219 1/20 0.34
RHEB Q15382 1/20 0.34
MMP2 P08253 1/20 0.34
MMP9 P14780 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926706 0.89 FLT1 (0.39) MEN1KMT2ACYP2C9CYP2C19ALDH1A1
SCHEMBL8925119 0.88 CA2 (0.43)
SCHEMBL8927101 0.87 CA2 (0.39)
SCHEMBL8926691 0.86 ALDH1A1 (0.36) CYP2C9CYP2C19ALDH1A1HTTL3MBTL1
SCHEMBL8925017 0.85 KDM4E (0.39) MEN1KMT2ACYP1A2CYP2C9CYP2C19
SCHEMBL7801836 0.83
SCHEMBL8925511 0.82 ALDH1A1 (0.38) ALDH1A1PTGS2
SCHEMBL27364824 0.81 SLC6A2 (0.41)
SCHEMBL8926714 0.79 PTGS1 (0.36) CYP2C9CYP2C19ALDH1A1HTTL3MBTL1
SCHEMBL8926788 0.78 PTGS2 (0.36) MEN1KMT2AALDH1A1MAPTPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US disclosed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN disclosed