SCHEMBL8925017

SCHEMBL8925017

Cc1cc(Sc2ccc(F)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
KCNQ3 O43525 1/20 0.36
KCNQ2 O43526 1/20 0.36
SLC9A1 P19634 1/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926231 0.88 RHEB (0.43) KDM4EALDH1A1MAPTHPGD
SCHEMBL8925113 0.87 CA12 (0.45) ALDH1A1HPGD
SCHEMBL8926370 0.86 SLC6A9 (0.36)
SCHEMBL8926916 0.86 PDE7A (0.41) PTGS2PTGS1SLC9A1
SCHEMBL8926718 0.85 AGBL2 (0.39) KDM4EALDH1A1MAPTHPGDPTGS2
SCHEMBL7798515 0.82 SLC9A1 (0.61) SLC9A1
SCHEMBL8927186 0.81 ALDH1A1 (0.40) ALDH1A1PTGS2SLC9A1
SCHEMBL8925087 0.80 PDE4B (0.41) MAPTHPGDMEN1KMT2A
SCHEMBL8926776 0.78 PTGS1 (0.38) PTGS2PTGS1
SCHEMBL8925101 0.77 ALDH1A1 (0.37) ALDH1A1MAPTHPGDPTGS2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US disclosed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN disclosed