SCHEMBL8926706

SCHEMBL8926706

CCc1cc(Sc2ccc(Cl)cc2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
PTGDR2 Q9Y5Y4 3/20 0.39
ALDH1A1 P00352 3/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA3 P07451 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8926718 0.89 AGBL2 (0.39) ALDH1A1CYP2C9CYP2C19KDM4EMAPT
SCHEMBL8925119 0.89 CA2 (0.43) CA12CA1CA2CA3CA4
SCHEMBL8926691 0.88 ALDH1A1 (0.36) ALDH1A1CYP2C9CYP2C19L3MBTL1CA12
SCHEMBL27364824 0.87 SLC6A2 (0.41) FLT1FLT4KDRCA12CA1
SCHEMBL8926231 0.85 RHEB (0.43) PTGDR2ALDH1A1KDM4ELMNAMAPT
SCHEMBL6932531 0.84
SCHEMBL8926788 0.81 PTGS2 (0.36) ALDH1A1LMNAMAPTHPGDCA12
SCHEMBL8927101 0.81 CA2 (0.39) CA12CA1CA2CA3CA4
SCHEMBL8926714 0.80 PTGS1 (0.36) ALDH1A1CYP2C9CYP2C19L3MBTL1CA12
SCHEMBL8926230 0.79 CA12 (0.32) CA12CA1CA2CA6CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN disclosed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US disclosed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN disclosed