SCHEMBL8927576

SCHEMBL8927576

COC(=O)CN(C(=O)C(NC(=O)OC(C)(C)C)[C@H](C)C(=O)O)C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.38
CTSK P43235 2/20 0.38
KMT2A Q03164 1/20 0.37
CACNA1B Q00975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7329222 0.82 CTSK (0.44) CTSSCTSK
SCHEMBL7337054 0.80 CTSL (0.43) CTSSCTSK
SCHEMBL7398209 0.79 CTSL (0.41) CTSSCTSK
SCHEMBL7564794 0.78 CTSL (0.41) CTSSCTSK
SCHEMBL10910692 0.77 CTSS (0.45) CTSSCTSKKMT2A
SCHEMBL3525420 0.74 EPHX2 (0.39)
SCHEMBL7572761 0.73 CTSL (0.40) CTSSCTSKKMT2A
SCHEMBL7025316 0.73 EPHX2 (0.36)
SCHEMBL4665948 0.72 CTSK (0.42) CTSSCTSKKMT2ACACNA1B
SCHEMBL5527345 0.72 CTSK (0.42) CTSSCTSKKMT2ACACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5677448-A CHEMICAL INTERMEDIATES FOR MAKING ANTAGONIST OF THROMBIN, TREATING THROMBOSIS, STROKE, INFLAMMATION, ARTERIOSCLEROSIS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-10-14 US disclosed
US-5405854-A Anticoagulants HOFFMANN-LA ROCHE INC. (US) 1995-04-11 US disclosed