SCHEMBL8928102

SCHEMBL8928102

COc1ccc(F)c(CCCNC(=O)C(C)C)c1

nearest known ligand 0.76

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 8/20 0.55
MTNR1A P48039 7/20 0.55
NQO2 P16083 2/20 0.53
KDM4E B2RXH2 1/20 0.50
TP53 P04637 1/20 0.50
MAPT P10636 1/20 0.50
ALOX15 P16050 1/20 0.50
HSD17B10 Q99714 1/20 0.50
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8928099 0.86 MTNR1B (0.73) MTNR1BMTNR1A
SCHEMBL8928098 0.82 MTNR1A (0.63) MTNR1A
SCHEMBL8928245 0.81 MTNR1A (0.56) MTNR1BMTNR1AKDM4EHSD17B10
SCHEMBL25335984 0.79 CYP2D6 (0.68) CYP2D6CYP2C9CYP2C19KMT2A
SCHEMBL8928123 0.77 MTNR1A (0.73) MTNR1BMTNR1ANQO2CYP2D6CYP2C9
SCHEMBL14430371 0.76 POLB (0.61) MTNR1BMTNR1AHSD17B10
SCHEMBL32684170 0.74 MTNR1A (0.63) MTNR1BMTNR1ANQO2KDM4ETP53
SCHEMBL793987 0.74 GLA (0.63) MTNR1BMTNR1AKMT2A
SCHEMBL8928133 0.74 MTNR1A (0.67) MTNR1BMTNR1ANQO2MAPTCYP2D6
SCHEMBL19304105 0.74 CHRM2 (0.54) MTNR1BMTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541228-A Melatonergic agents BRISTOL-MYERS SQUIBB CO. (US) 1996-07-30 US claimed
EP-0706994-A1 Melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-17 EP claimed
US-5661185-A AN ALKOXYPHENYL-ALKYLUREA COMPOUND TREATING SLEEP DISORDER BRISTOL-MYERS SQUIBB CO. (US) 1997-08-26 US disclosed
US-5597651-A Rubber-polyester composites including polystyrene-polyester copolymers HOECHST CELANESE CORP. (US) 1997-01-28 US disclosed
US-5541228-A Melatonergic agents BRISTOL-MYERS SQUIBB CO. (US) 1996-07-30 US disclosed
EP-0706994-A1 Melatonergic agents BRISTOL-MYERS SQUIBB COMPANY (US) 1996-04-17 EP disclosed