SCHEMBL8928246

SCHEMBL8928246

CC1=C(C#N)C(c2cccc(-n3ccnc3)c2)C(C#N)=C(C)N1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.44
CYP3A4 P08684 4/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
GAA P10253 1/20 0.41
CYP11B1 P15538 2/20 0.38
CYP11B2 P19099 2/20 0.38
CYP19A1 P11511 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
MET P08581 1/20 0.38
CYP2A6 P11509 1/20 0.38
F10 P00742 1/20 0.37
PDE2A O00408 2/20 0.37
PDE1A P54750 2/20 0.37
PDE1B Q01064 2/20 0.37
PDE3B Q13370 2/20 0.37
PDE1C Q14123 2/20 0.37
PDE3A Q14432 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8860432 0.86 POLB (0.49) IDO1CYP3A4CYP1A2CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8928281 0.85 POLB (0.48) IDO1CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL8782154 0.79 IDO1 (0.47) IDO1CYP3A4GAA
SCHEMBL8928255 0.79 CHRNA7 (0.44) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8928204 0.76 CACNA1C (0.40) IDO1GAAPDE2APDE1APDE1B
SCHEMBL8928277 0.73 CACNA1C (0.54) CYP3A4CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL13295967 0.72 ALDH1A1 (0.53) GAALMNAMAPT
SCHEMBL8928241 0.72 KDM4E (0.53) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL13295965 0.71 CUL4A (0.53) CYP3A4CYP1A2CYP2C9CYP2C19GAA
SCHEMBL31420979 0.70 IDO1 (0.58) IDO1CYP3A4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP claimed
EP-0755931-A1 Dihydropyridine and pyridine derivatives and process for their preparation PHARMACIA & UPJOHN S.p.A. (IT) 1997-01-29 EP disclosed