SCHEMBL8928685

SCHEMBL8928685

O=C(Cl)Cc1cc2ccccc2[nH]1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 1/20 0.55
NLRP3 Q96P20 1/20 0.54
MTNR1A P48039 1/20 0.53
MTNR1B P49286 1/20 0.53
FLT3 P36888 1/20 0.50
IDO1 P14902 2/20 0.49
KDM4E B2RXH2 2/20 0.49
DAO P14920 2/20 0.49
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
SRD5A2 P31213 1/20 0.49
HSD17B10 Q99714 1/20 0.49
SIRT1 Q96EB6 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.47
GSK3B P49841 1/20 0.45
HDAC3 O15379 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC2 Q92769 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29966882 1.00 LOXL2 (0.55) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL3451201 0.85 LOXL2 (0.58) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL29365671 0.84 LOXL2 (0.56) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL31336079 0.84 LOXL2 (0.56) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL49270 0.84 LOXL2 (0.56) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL3120573 0.82 MTNR1A (0.60) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL630523 0.82 SIRT1 (0.64) LOXL2NLRP3MTNR1AMTNR1BFLT3
Water SCHEMBL30025993 0.82 LOXL2 (0.55) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL31511816 0.82 LOXL2 (0.55) LOXL2NLRP3MTNR1AMTNR1BFLT3
SCHEMBL3447317 0.82 LOXL2 (0.55) LOXL2NLRP3MTNR1AMTNR1BFLT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776892-A1 THIENYLAZOLE COMPOUND AND THIENOTRIAZOLODIAZEPINE COMPOUND YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-06-04 EP disclosed
US-4563464-A 2-Azabicyclo(2.2.2)octane derivatives and their use as immunosuppressive agents RICHTER GEDEON VEGYESZETI GYAR RT. (HU) 1986-01-07 US disclosed
EP-0132964-A2 2-Azabicyclo[2.2.2]octane derivatives RICHTER GEDEON VEGYESZETI GYAR R.T. (HU) 1985-02-13 EP disclosed