SCHEMBL8930729

SCHEMBL8930729

CCN(CC)C(=O)c1c2c(c(C(c3c4c(cc5c3OC(C)(C)O5)OC(C)(C)O4)c3c4c(c(C(=O)N(CC)CC)c5c3OC(C)(C)O5)OC(C)(C)O4)c3c1OC(C)(C)O3)OC(C)(C)O2

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
HSP90AA1 P07900 4/20 0.33
HSP90AB1 P08238 4/20 0.33
HTT P42858 1/20 0.32
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
HASPIN Q8TF76 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
HPGD P15428 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
KMT2A Q03164 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8930681 0.90 TSHR (0.34) TSHRHSP90AA1HSP90AB1HTTLMNA
SCHEMBL9273756 0.77 TSHR (0.36) TSHRHPGDALDH1A1
SCHEMBL8930666 0.77 TSHR (0.36) TSHRHSP90AA1HSP90AB1HTTSMN1; SMN2
SCHEMBL8930676 0.68 PTPN1 (0.33) ALDH1A1
SCHEMBL8930717 0.67 ALDH1A1 (0.39) SMN1; SMN2HPGDMEN1LMNAKMT2A
Tromethamine SCHEMBL9719398 0.67 TSHR (0.35) TSHRSMN1; SMN2HPGDMEN1LMNA
SCHEMBL7519849 0.65 TSHR (0.50) TSHRSMN1; SMN2HPGDALDH1A1
SCHEMBL7514575 0.64 CYP3A4 (0.45) TSHRSMN1; SMN2HPGDMEN1KMT2A
SCHEMBL7514564 0.61 TSHR (0.45) TSHRHTTCCNCCDK8SMN1; SMN2
SCHEMBL8930638 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5599522-A CONTRAST ENHANCING AGENTS NYCOMED IMAGING AS (NO) 1997-02-04 US disclosed
EP-0515458-B1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI NYCOMED INNOVATION AB (SE) 1995-08-23 EP disclosed
EP-0515458-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI. HAFSLUND NYCOMED INNOVATION (SE) 1992-12-02 EP disclosed
WO-1991012024-A1 TRIARYLMETHYL RADICALS AND THE USE OF INERT CARBON FREE RADICALS IN MRI HAFSLUND NYCOMED INNOVATION AB (SE) 1991-08-22 WO disclosed