SCHEMBL8933495

SCHEMBL8933495

COC(CNC1=Nc2ccc(C#N)cc2C(c2ccccc2F)=NC1)OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA3 P34903 5/20 0.41
GABRA5 P31644 4/20 0.41
GABRA1 P14867 3/20 0.41
GABRA2 P47869 3/20 0.41
GABRB2 P47870 2/20 0.41
CCNE2 O96020 1/20 0.39
EGFR P00533 1/20 0.39
CDK1 P06493 1/20 0.39
CDK4 P11802 1/20 0.39
SRC P12931 1/20 0.39
CCND1 P24385 1/20 0.39
CCNE1 P24864 1/20 0.39
CDK2 P24941 1/20 0.39
KDR P35968 1/20 0.39
CCNA1 P78396 1/20 0.39
PTK2 Q05397 1/20 0.39
GABRG2 P18507 4/20 0.37
GABRB3 P28472 4/20 0.37
PTAFR P25105 6/20 0.33
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8933416 0.82 GABRA3 (0.35) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11833620 0.80 GABRA5 (0.44) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL14217666 0.76 GABRA1 (0.55) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL7415888 0.74 GABRA3 (0.47) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11827503 0.73 GABRA1 (0.45) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11830651 0.71 GABRA3 (0.42) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11158188 0.71 TP53 (0.39) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11827831 0.70 GABRA1 (0.48) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11826182 0.69 GABRA1 (0.47) GABRA3GABRA5GABRA1GABRA2GABRB2
SCHEMBL11826517 0.69 CHRM1 (0.47) GABRA3GABRA5GABRA1GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996023790-A1 ACETYLIMIDAZOBENZODIAZEPINES F. HOFFMANN-LA ROCHE AG (CH) 1996-08-08 WO disclosed